2,5-disubstituted bicyclo[2.1.1]hexanes as rigidified cyclopentane variants

نویسندگان

چکیده

Identification of rigid counterparts for common flexible scaffolds is crucial to the advancement medicinal chemistry. Herein, synthesis new bicyclo[2.1.1]hexanes act as rigidified cyclopentanes described.

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ژورنال

عنوان ژورنال: Chemical Science

سال: 2023

ISSN: ['2041-6520', '2041-6539']

DOI: https://doi.org/10.1039/d3sc02695g